Mianserin hydrochloride ( Mianserin hydrochloride; Tolvon; Tolvin; ORG GB 94; Lerivon )

产品货号. M13439 CAS No. 21535-47-7

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Mianserin hydrochloride
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Mianserin hydrochloride is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
产品描述

Mianserin hydrochloride is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
同义词

Mianserin hydrochloride; Tolvon; Tolvin; ORG GB 94; Lerivon
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

5-HT; HT; Sert (Sodium-dependent); Adrenergic Receptor; DA transporter; Dopamine; Noradrenaline transporter (Sodium-dependent)κ-opioid receptor
研究领域

Neurological Disease
适应症

——

CAS Number

21535-47-7
分子量

300.83
分子式

C18H21ClN2
纯度

>98%(HPLC)
溶解度

Ethanol: 21 mg/mL (69.8 mM); Water: 30 mg/mL (99.72 mM); DMSO: 60 mg/mL (199.44 mM)
SMILES

CN1CCN2C(C1)C3=CC=CC=C3CC4=CC=CC=C42.Cl
化学全称

2-methyl-1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyrazino[1,2-a]azepine hydrochloride

1.Dekeyne A, Millan MJ. Neuropharmacology. 2006 Sep;51(4):718-26.

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